SCHEMBL28197938

SCHEMBL28197938

OCc1ccc(-c2ccn(O)n2)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
EGFR P00533 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
KDM1A O60341 1/20 0.32
HDAC1 Q13547 1/20 0.32
DHODH Q02127 1/20 0.32
CSNK1D P48730 1/20 0.31
CSNK1E P49674 1/20 0.31
PDK2 Q15119 1/20 0.31
RORC P51449 1/20 0.31
GRM2 Q14416 3/20 0.31
ACSS2 Q9NR19 1/20 0.31
CYP2C9 P11712 1/20 0.30
HSD17B10 Q99714 1/20 0.30
KIF11 P52732 1/20 0.30
PDE4B Q07343 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5650249 0.73 IDO1 (0.42)
SCHEMBL877208 0.68 GRM2 (0.47) CYP4F2CYP4A11GRM2CYP2C9S1PR3
SCHEMBL538836 0.67 PTGS1 (0.47) KMT2APDK2CYP2C9
SCHEMBL25792021 0.67 CYP1A2 (0.36) P2RX7HDAC1DHODHCSNK1DCSNK1E
SCHEMBL28198655 0.67 CYP11B2 (0.41) S1PR1
SCHEMBL93021 0.65 CYP4F2 (0.50) CYP4F2CYP4A11KIF11
SCHEMBL15725317 0.65 BACE1 (0.46) CYP4F2CYP4A11KIF11S1PR1PRKAB2
SCHEMBL19568037 0.64 ACSS2 (0.36) KMT2AKDM1AHDAC1PDK2GRM2
SCHEMBL22143054 0.63 USP1 (0.43) P2RX7HDAC1KIF11
SCHEMBL15725334 0.62 RARB (0.52) CYP4F2CYP4A11HSD17B10KIF11S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107667106-A 2 (base of Pyrazolopyridine 3) pyrimidine derivatives as JAK inhibitor 阿尔米雷尔有限公司 2018-02-06 CN disclosed