SCHEMBL28199583

SCHEMBL28199583

O=CNc1ccnc(-c2ccc(F)c(F)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 5/20 0.44
TGFBR1 P36897 3/20 0.41
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38
EGLN2 Q96KS0 1/20 0.37
PPARG P37231 1/20 0.36
CNR1 P21554 1/20 0.35
TOP1 P11387 1/20 0.35
NOTUM Q6P988 1/20 0.35
MAOB P27338 1/20 0.35
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
WNT3A P56704 1/20 0.33
CYP17A1 P05093 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28856056 0.84 PPARG (0.47) TGFBR1RAB9AALDH1A1MAPK1CYP1A2
SCHEMBL3905856 0.78 KMO (0.47) KMORAB9AKDM4EALDH1A1MAPK1
SCHEMBL28200272 0.78 HDAC1 (0.50) TGFBR1TOP1MAPKAPK2
SCHEMBL28856181 0.75 LOXL2 (0.50) TGFBR1PPARGCNR1
SCHEMBL241795 0.74 RAB9A (0.46) RAB9AALDH1A1NPC1MAPTNFKB1
SCHEMBL28200295 0.74 KDM2B (0.38) CNR1NOTUM
SCHEMBL2666352 0.70 CCR1 (0.57) KMORAB9AKDM4EALDH1A1MAPK1
SCHEMBL4120500 0.70 CYP11B1 (0.46) KMORAB9AKDM4EALDH1A1MAPK1
SCHEMBL3904494 0.69 CYP11B1 (0.45) KMORAB9AKDM4EALDH1A1MAPK1
SCHEMBL28199585 0.68 KMO (0.52) KMORAB9AKDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107709311-A The carboxamides derivatives of 2 phenyl, 6 imidazolyl pyridines 4 and its purposes as EAAT3 inhibitor 豪夫迈·罗氏有限公司 2018-02-16 CN disclosed