SCHEMBL28199804

SCHEMBL28199804

CC(C)c1ccc(Nc2cncc(C(N)=O)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
KIF11 P52732 1/20 0.43
ALDH1A1 P00352 3/20 0.42
NFKB1 P19838 2/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
CDK2 P24941 2/20 0.41
SMN1; SMN2 Q16637 5/20 0.40
KCNH2 Q12809 2/20 0.40
SCN5A Q14524 2/20 0.40
SCN9A Q15858 2/20 0.40
TP53 P04637 2/20 0.40
LMNA P02545 1/20 0.40
P2RX3 P56373 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469190 0.74 MAPK1 (0.43) ALDH1A1
SCHEMBL19151634 0.69 ADORA3 (0.42) KCNH2SCN9ALMNA
SCHEMBL31636273 0.69 ADORA3 (0.42) KCNH2SCN9ALMNA
SCHEMBL19447116 0.69 CSF1R (0.53)
SCHEMBL5042271 0.68 HCAR3 (0.39) GAALMNAMEN1KMT2AL3MBTL1
SCHEMBL2789615 0.68 RAB9A (0.64) NPC1RAB9AALDH1A1NFKB1CDK2
SCHEMBL6468902 0.68 FYN (0.46) CDK2KCNH2SCN9AP2RX3
SCHEMBL7109264 0.67 TSHR (0.56) ALDH1A1KCNH2LMNAKMT2A
SCHEMBL23080875 0.66 NPC1 (0.44) NPC1RAB9AKIF11ALDH1A1NFKB1
SCHEMBL27987796 0.66 MAP3K14 (0.47) SCN9ABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107709315-A The inhibitor of bruton's tyrosine kinase 药品循环有限责任公司 2018-02-16 CN disclosed