SCHEMBL28201512

SCHEMBL28201512

Cn1cc2cc(C(N)=O)ccc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.54
MAOB P27338 3/20 0.54
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 2/20 0.46
BRD4 O60885 1/20 0.46
BRPF1 P55201 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NSD2 O96028 1/20 0.45
MAPT P10636 1/20 0.45
DYRK1A Q13627 1/20 0.44
LCK P06239 1/20 0.43
KMT2A Q03164 1/20 0.42
NOTUM Q6P988 1/20 0.41
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
STING1 Q86WV6 1/20 0.41
CHEK2 O96017 2/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28856319 0.98 MAOA (0.53) MAOAMAOBKDM4EALDH1A1BRD4
Formic Acid SCHEMBL30427064 0.94 MAOA (0.50) MAOAMAOBKDM4EALDH1A1BRD4
SCHEMBL9989118 0.87 KDM4E (0.57) MAOAMAOBKDM4EALDH1A1BRD4
SCHEMBL1144800 0.85 MAOA (0.56) MAOAMAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL28591105 0.85 MAOA (0.59) MAOAMAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL26170012 0.83 MAOA (0.58) MAOAMAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL1144873 0.81 MAOA (0.55) MAOAMAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL28037046 0.81 MAOA (0.52) MAOAMAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL30177194 0.80 HPGDS (0.40) MAOAMAOBKDM4EALDH1A1BRD4
SCHEMBL12073303 0.79 MAP2K4 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551593-A Compounds and methods for modulating splicing 雷密克斯医疗公司 2022-12-30 CN disclosed
CN-105451737-B Medical composition and its use and described pharmaceutical composition are used for the application process practised contraception on demand 拜耳医药股份有限公司 2018-04-10 CN disclosed