SCHEMBL28201879

SCHEMBL28201879

Cc1nccc(COCc2ccnc(C)c2C)c1C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.33
MAOA P21397 2/20 0.32
DCPS Q96C86 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10647777 0.85 DYRK1A (0.40) CYP2A6MAOADYRK1A
SCHEMBL3801869 0.77 NOS2 (0.38) CYP2A6NOS3NOS2
SCHEMBL1931165 0.76 LOXL2 (0.45) CYP2A6NOS3NOS2
SCHEMBL4795960 0.76 KDM4E (0.41) CYP2A6MAOANOS3NOS2DYRK1A
SCHEMBL156074 0.76 CYP2A6 (0.34) CYP2A6NOS3NOS2
SCHEMBL7396568 0.76 CYP2A6 (0.34) CYP2A6NOS3NOS2
SCHEMBL25820190 0.72 GABRA1 (0.38) CYP2A6MAOANOS3NOS2
SCHEMBL11500900 0.71 CYP2D6 (0.37) DYRK1A
SCHEMBL27570675 0.71 TYR (0.37) NOS2DYRK1A
SCHEMBL7696876 0.71 CYP2A6 (0.31) CYP2A6MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106146349-B A kind of method that aromatic aldehyde catalyzed conversion prepares amidine 中国科学院大连化学物理研究所 2018-02-13 CN disclosed