SCHEMBL28202151

SCHEMBL28202151

O=CNc1cnc2cncc(CC(F)(F)F)c2c1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.34
ROCK2 O75116 2/20 0.34
JAK1 P23458 2/20 0.34
TYK2 P29597 2/20 0.34
JAK3 P52333 2/20 0.34
ROCK1 Q13464 2/20 0.34
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
JAK2 O60674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28058293 0.71 HPGDS (0.35) IKBKBROCK2JAK1TYK2JAK3
SCHEMBL28202148 0.71 GSK3A (0.42) ROCK2CDK2
SCHEMBL28202187 0.71 F10 (0.34) ROCK1CDK2
SCHEMBL28202753 0.70 DYRK1A (0.40) CDK2
SCHEMBL28202190 0.69 ERN1 (0.35)
SCHEMBL28202183 0.68 ERN1 (0.36)
SCHEMBL28202145 0.65 F2RL3 (0.34)
SCHEMBL27918809 0.64 ALDH1A1 (0.44)
SCHEMBL28170955 0.63 NPC1 (0.41)
SCHEMBL24628752 0.60 ALDH1A1 (0.46) CCNE2CDK4CCND1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473568-B 1, 7-naphthyridine derivatives 豪夫迈·罗氏有限公司 2018-02-13 CN disclosed