SCHEMBL28058293

SCHEMBL28058293

NC(=O)c1cnc2cncc(CC(F)(F)F)c2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.35
NNMT P40261 5/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CDK1 P06493 1/20 0.32
PIM1 P11309 1/20 0.32
CDK2 P24941 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
DYRK1A Q13627 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
MAP4K4 O95819 1/20 0.31
PSMD14 O00487 1/20 0.31
STAMBP O95630 1/20 0.31
COPS5 Q92905 1/20 0.31
IKBKB O14920 1/20 0.31
ROCK2 O75116 1/20 0.31
JAK1 P23458 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16438181 0.75 ALPL (0.42) HPGDSNNMTDYRK1ASIRT2SIRT1
SCHEMBL840723 0.75 NNMT (0.36) HPGDSNNMTSMN1; SMN2PSMD14STAMBP
SCHEMBL28058331 0.75 HPGDS (0.33) HPGDSNNMTCYP11B1CYP11B2
SCHEMBL17755580 0.73 HPGDS (0.39) HPGDSNNMTSMN1; SMN2CYP11B1CYP11B2
SCHEMBL28202150 0.73 HPGDS (0.40) HPGDSNNMTSMN1; SMN2MAP4K4PSMD14
SCHEMBL16432565 0.73 HPGDS (0.40) HPGDSNNMTSMN1; SMN2MAP4K4PSMD14
SCHEMBL18783466 0.72 MKNK1 (0.40) HPGDSNNMTSMN1; SMN2CYP11B1CYP11B2
SCHEMBL28202151 0.71 IKBKB (0.34) CDK2IKBKBROCK2JAK1TYK2
SCHEMBL28229692 0.71 CYP11B2 (0.45) CYP11B1CYP11B2KDM4EMKNK1MKNK2
SCHEMBL16432422 0.71 MAP4K4 (0.44) CDK1PIM1CDK2MAPKAPK2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473568-B 1, 7-naphthyridine derivatives 豪夫迈·罗氏有限公司 2018-02-13 CN disclosed
CN-105473568-A 1, 7-naphthyridine derivatives HOFFMANN LA ROCHE 2016-04-06 CN disclosed