SCHEMBL28210277

SCHEMBL28210277

O=C(O)NNc1cc(CO)nn1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
LMNA P02545 4/20 0.50
NTRK1 P04629 2/20 0.47
GAA P10253 1/20 0.44
KCNJ6 P48051 5/20 0.43
KCNJ5 P48544 5/20 0.43
KCNJ3 P48549 5/20 0.43
TSHR P16473 1/20 0.43
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA9 Q16790 3/20 0.42
HTT P42858 2/20 0.42
PTGS2 P35354 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ATM Q13315 1/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
STAT1 P42224 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16780330 0.85 ALDH1A1 (0.59) ALDH1A1LMNANTRK1GAAKCNJ6
SCHEMBL27954241 0.84 FAAH (0.49) ALDH1A1LMNANTRK1GAAKCNJ6
SCHEMBL27767837 0.84 ALDH1A1 (0.58) ALDH1A1LMNANTRK1GAAKCNJ6
SCHEMBL2837900 0.79 GAA (0.67) ALDH1A1LMNAGAAMEN1KMT2A
SCHEMBL2839406 0.78 GAA (0.60) ALDH1A1LMNAGAAKCNJ6KCNJ5
SCHEMBL13858692 0.76 FAAH (0.51) ALDH1A1LMNANTRK1GAAKCNJ6
SCHEMBL2837826 0.75 ALDH1A1 (0.57) ALDH1A1LMNATSHRCA1CA2
SCHEMBL16804455 0.73 MAPT (0.63) ALDH1A1GAACA1CA2CA9
SCHEMBL17361370 0.73 PTGS2 (0.49) ALDH1A1LMNAGAACA1CA2
SCHEMBL27767901 0.73 LMNA (0.46) ALDH1A1LMNANTRK1KCNJ6KCNJ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903310-B Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain 阵列生物制药公司 2018-08-14 CN disclosed
CN-108329246-A Pyrrolidinyl urea and pyrrolidinyl thiourea compound as TRKA kinase inhibitors 阵列生物制药公司 2018-07-27 CN disclosed
CN-105130967-B Pyrrolidinyl urea and pyrrolidinyl thiourea compound as TRKA kinase inhibitors 阵列生物制药公司 2018-04-17 CN disclosed