SCHEMBL2821301

SCHEMBL2821301

c1cc(-c2ccc(C34CCCN(CC3)C4)nn2)co1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.35
KCNH2 Q12809 1/20 0.35
PBRM1 Q86U86 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 2/20 0.33
ALOX15 P16050 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL668390 0.82 ACHE (0.36) ALDH1A1
SCHEMBL5220727 0.81 CYP11B1 (0.38) CHRNA7KCNH2ALDH1A1CYP1A2ALOX15
Bromide SCHEMBL4482662 0.80 CYP11B1 (0.37) CHRNA7KCNH2ALDH1A1CYP1A2ALOX15
SCHEMBL2820263 0.79 SLC6A2 (0.31)
SCHEMBL2677748 0.78 CYP11B1 (0.39) CHRNA7KCNH2ALDH1A1CYP1A2ALOX15
SCHEMBL2823249 0.78 ALDH1A1 (0.39) PBRM1ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL2823335 0.78 SLC6A2 (0.30)
SCHEMBL2819737 0.77 SCD (0.35)
Hydrochloric Acid SCHEMBL2819670 0.77 ALDH1A1 (0.38) PBRM1ALDH1A1HSD17B10
SCHEMBL2819424 0.77 KCNH2 (0.36) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922320-B1 DERIVATIVES OF 5-PYRIDAZINYL-1-AZABICYCLO[3.2.1]OCTANE, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2010-10-27 EP claimed