SCHEMBL2822113

SCHEMBL2822113

COc1ccc(-c2ccc(C34CCCN(CC3)C4)nn2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
HPGD P15428 4/20 0.43
MAPK1 P28482 3/20 0.43
POLB P06746 3/20 0.43
MAPT P10636 4/20 0.41
USP2 O75604 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 3/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
PKM P14618 2/20 0.39
TP53 P04637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
BRD4 O60885 1/20 0.39
ALOX15 P16050 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2822814 0.99 ALDH1A1 (0.42) ALDH1A1HPGDMAPK1POLBMAPT
SCHEMBL2818964 0.85 NPC1 (0.41) MAPTKMT2AMEN1GAAKDM4E
Hydrochloric Acid SCHEMBL2824030 0.84 NPC1 (0.40) MAPTKMT2AMEN1GAAKDM4E
SCHEMBL5223011 0.82 FYN (0.40) ALDH1A1HPGDMAPK1POLBUSP2
Bromide SCHEMBL4460701 0.81 FYN (0.40) ALDH1A1HPGDMAPK1POLBUSP2
SCHEMBL2820263 0.80 SLC6A2 (0.31)
SCHEMBL2678759 0.79 FYN (0.42) ALDH1A1HPGDMAPK1POLBMAPT
Hydrochloric Acid SCHEMBL2823335 0.79 SLC6A2 (0.30)
Hydrochloric Acid SCHEMBL2678564 0.78 FYN (0.41) ALDH1A1HPGDMAPK1POLBMAPT
SCHEMBL668390 0.78 ACHE (0.36) ALDH1A1MAPTUSP2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922320-B1 DERIVATIVES OF 5-PYRIDAZINYL-1-AZABICYCLO[3.2.1]OCTANE, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2010-10-27 EP claimed