SCHEMBL28223333

SCHEMBL28223333

CCCc1cc(C#N)ccc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
MTOR P42345 1/20 0.41
GSK3B P49841 1/20 0.41
PRKDC P78527 1/20 0.41
KCNH2 Q12809 1/20 0.41
ATM Q13315 1/20 0.41
ATR Q13535 1/20 0.41
CASP1 P29466 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPK8 P45983 2/20 0.37
PARP1 P09874 1/20 0.37
PARP15 Q460N3 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11434090 0.86 XDH (0.43) MEN1KMT2AABCC9ABCC8KCNJ11
SCHEMBL5479625 0.81 NPC1 (0.49)
SCHEMBL7409664 0.77 PRKCI (0.40) KDRKCNH2CASP1MEN1KMT2A
SCHEMBL2977013 0.77 HSD17B10 (0.42) KDRMEN1KMT2APARP1PARP10
SCHEMBL22067721 0.77 MAPK8 (0.39) KDRMEN1KMT2AMAPK8PARP1
SCHEMBL12663273 0.76 CYP2A6 (0.45) KDRHRH4MEN1KMT2AABCC9
SCHEMBL14291553 0.76 CYP2A6 (0.45) KDRHRH4MEN1KMT2AABCC9
SCHEMBL5483765 0.76 DGAT1 (0.51) KDRCASP1MEN1KMT2APARP1
SCHEMBL28252825 0.76 FLT1 (0.56) KDRCASP1MEN1KMT2AADRA1D
SCHEMBL28222517 0.76 LMNA (0.46) MEN1KMT2AMAPK8PARP1PARP15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105399685-B The alternatively preparation method and applications of the heteroaromatic compounds of property JAK3 and/or JAK1 kinase inhibitors 深圳微芯生物科技有限责任公司 2018-05-22 CN disclosed