SCHEMBL282248

SCHEMBL282248

CCOP(=O)(OCC)C(N)P(=O)(OCC)OCC

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PPARD Q03181 2/20 0.37
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
LAP3 P28838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405218 0.85 LAP3 (0.44) TSHRTP53TDP1POLBCYP3A4
SCHEMBL14064086 0.81 TSHR (0.46) TSHRTP53TDP1POLBCYP3A4
SCHEMBL3175484 0.81 TSHR (0.46) TSHRTP53TDP1POLBCYP3A4
SCHEMBL18946366 0.81 TSHR (0.46) TSHRTP53TDP1POLBCYP3A4
SCHEMBL492011 0.79 LAP3 (0.48) TSHRTP53TDP1POLBCYP3A4
SCHEMBL9157801 0.77 LAP3 (0.42) TSHRTP53TDP1POLBCYP3A4
SCHEMBL10911354 0.77 TSHR (0.53) TSHRTP53TDP1POLBCYP3A4
SCHEMBL4402436 0.75 TSHR (0.40) TSHRTP53TDP1POLBCYP3A4
SCHEMBL28659627 0.75 TSHR (0.40) TSHRTP53TDP1POLBCYP3A4
SCHEMBL10201143 0.74 TSHR (0.50) TSHRTP53TDP1POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9828393-B2 Silylalkyloxyaryl compounds and methods for treating cancer THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2017-11-28 US claimed
US-20160159832-A1 SILYLALKYLOXYARYL COMPOUNDS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE 2016-06-09 US claimed
WO-2015013322-A1 SILYLALKYLOXYARYL COMPOUNDS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2015-01-29 WO claimed
WO-2025024714-A2 BONE-TARGETED CANONICAL NOTCH INHIBITOR BIOVENTURES, LLC (US) 2025-01-30 WO disclosed
US-20230330116-A1 MATERIALS AND METHODS FOR SUPPRESSING AND/OR TREATING BONE RELATED DISEASES AND SYMPTOMS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2023-10-19 US disclosed
US-11672811-B2 Materials and methods for suppressing and/or treating bone related diseases and symptoms INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2023-06-13 US disclosed
US-11497813-B2 Bortezomib conjugates and methods using same BIOVINC, LLC (US) 2022-11-15 US disclosed
US-11497813-B2 Bortezomib conjugates and methods using same BIOVINC, LLC (US) 2022-11-15 US disclosed
US-20220125959-A1 PROSTATE-SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS AS DIAGNOSTIC AND RADIONUCLIDE THERAPEUTIC AGENTS FIVE ELEVEN PHARMA INC (US) 2022-04-28 US disclosed
US-20200368259-A1 MATERIALS AND METHODS FOR SUPPRESSING AND/OR TREATING BONE RELATED DISEASES AND SYMPTOMS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2020-11-26 US disclosed
WO-2020220023-A1 PROSTATE-SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS AS DIAGNOSTIC AND RADIONUCLIDE THERAPEUTIC AGENTS FIVE ELEVEN PHARMA INC. (US) 2020-10-29 WO disclosed
EP-0546548-B1 Guanidinyl alkyl-1,1-bis phosphonic acid derivatives, process for their preparation and their use HOECHST AG (DE) 1997-05-02 EP disclosed
EP-0531253-B1 N-substituted aminomethanediphosphonic acids CIBA GEIGY AG (CH) 1997-01-08 EP disclosed
US-5457094-A Bone disorder CIBA-GEIGY CORPORATION (US) 1995-10-10 US disclosed
US-5413994-A Some of the amidines as new compounds; use as calcium metabolism regulators CIBA-GEIGY CORPORATION (US) 1995-05-09 US disclosed
US-5294608-A Compounds for treatment of osteoporosis and bone disorders HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-15 US disclosed
US-5281748-A N-substituted aminomethanediphosphonic acids CIBA-GEIGY CORP. (US) 1994-01-25 US disclosed
EP-0555845-A2 Steroid derivatives MITSUBISHI KASEI CORPORATION (JP) 1993-08-18 EP disclosed
EP-0546548-A1 Guanidinyl alkyl-1,1-bis phosphonic acid derivatives, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-06-16 EP disclosed
EP-0531253-A1 N-substituted aminomethanediphosphonic acids CIBA-GEIGY AG (CH) 1993-03-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200368259-A1 MATERIALS AND METHODS FOR SUPPRESSING AND/OR TREATING BONE RELATED DISEASES AND SYMPTOMS SOST, TSG101, BST2 TSHR 4492/4885TP53 430/4885TDP1 3096/4885
US-11672811-B2 Materials and methods for suppressing and/or treating bone related diseases and symptoms SOST, TSG101, BST2 TSHR 4492/4885TP53 430/4885TDP1 3096/4885
US-20160159832-A1 SILYLALKYLOXYARYL COMPOUNDS AND METHODS FOR TREATING CANCER BCL3, MYLK2, BCL2L13 TSHR 4239/4885TP53 122/4885TDP1 4243/4885
US-11497813-B2 Bortezomib conjugates and methods using same BCR, PSMA6, PSMA5 TSHR 4516/4885TP53 505/4885TDP1 4145/4885
US-20220125959-A1 PROSTATE-SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS AS DIAGNOSTIC AND RADIONUCLIDE THERAPEUTIC AGENTS KLK3, FOLH1, PSMA1 TSHR 2054/4885TP53 473/4885TDP1 3910/4885
US-20230330116-A1 MATERIALS AND METHODS FOR SUPPRESSING AND/OR TREATING BONE RELATED DISEASES AND SYMPTOMS SOST, TSG101, ACP3 TSHR 4485/4885TP53 388/4885TDP1 3080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.