SCHEMBL28227656

SCHEMBL28227656

Brc1cccc(Cn2c(-c3cccc(Br)c3)nc3ccccc32)c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.77
LMNA P02545 2/20 0.77
TP53 P04637 6/20 0.70
TSHR P16473 1/20 0.67
HSD17B10 Q99714 1/20 0.67
HTT P42858 2/20 0.65
ALDH1A1 P00352 4/20 0.65
PDE6D O43924 1/20 0.65
ALDH2 P05091 1/20 0.65
ALDH3A1 P30838 1/20 0.65
CFTR P13569 1/20 0.62
HDAC1 Q13547 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
GALR3 O60755 1/20 0.53
NR2F2 P24468 1/20 0.53
TNF P01375 1/20 0.51
NPSR1 Q6W5P4 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15568415 0.87 MAPT (1.00) MAPTLMNATP53TSHRHSD17B10
SCHEMBL6562002 0.85 GALR3 (0.74) MAPTLMNATP53TSHRHSD17B10
SCHEMBL30934017 0.83 MAPT (0.80) MAPTLMNATP53TSHRHSD17B10
SCHEMBL29076181 0.83 MAPT (0.67) MAPTLMNATP53TSHRHSD17B10
SCHEMBL30581242 0.83 MAPT (0.67) MAPTLMNATP53TSHRHSD17B10
SCHEMBL28322548 0.81 TP53 (0.71) MAPTLMNATP53TSHRHTT
SCHEMBL29412044 0.81 TP53 (1.00) MAPTLMNATP53TSHRHSD17B10
SCHEMBL29412062 0.80 TP53 (0.78) MAPTLMNATP53HTTALDH1A1
SCHEMBL229828 0.79 ALDH1A1 (1.00) MAPTLMNATP53TSHRHSD17B10
SCHEMBL20797646 0.79 MYC (0.63) MAPTLMNATP53TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250202-B 2,3- disubstituted benzenes and imidazo [1,2-a] pyrimidines and its preparation method and application 陕西师范大学 2019-10-25 CN disclosed
CN-108250202-A 2,3- disubstituted benzenes and imidazo [1,2-a] pyrimidines and its preparation method and application 陕西师范大学 2018-07-06 CN disclosed