SCHEMBL28229161

SCHEMBL28229161

C=CCOc1cnccc1N

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.41
GAA P10253 1/20 0.38
POLB P06746 1/20 0.38
TGFBR1 P36897 1/20 0.37
TGFBR2 P37173 1/20 0.37
AOC1 P19801 2/20 0.36
AOC3 Q16853 2/20 0.36
TSHR P16473 2/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2A6 P11509 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13345451 0.86 IMPDH2 (0.41) IMPDH2GAAPOLBTGFBR1TGFBR2
SCHEMBL3823546 0.83 POLB (0.43) GAAPOLBTGFBR1TGFBR2TSHR
SCHEMBL4956799 0.79 ADRA2A (0.40) GAAPOLBTGFBR1TGFBR2TSHR
SCHEMBL2790469 0.76 GAA (0.42) IMPDH2GAAAOC1AOC3CYP3A4
SCHEMBL11628534 0.76 ALDH1A1 (0.53) GAAPOLBAOC1AOC3HPGD
SCHEMBL8811300 0.75 POLB (0.38) GAAPOLBTGFBR1TGFBR2TSHR
SCHEMBL15288914 0.73 GAA (0.52) GAATSHRMAPT
SCHEMBL4958013 0.73 POLB (0.40) GAAPOLBTGFBR1TGFBR2HPGD
SCHEMBL4608367 0.73 ALDH1A1 (0.55) TSHRHPGDMAPK1HSD17B10CYP3A4
SCHEMBL27624925 0.73 ALDH1A1 (0.47) GAAPOLBAOC1AOC3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191781-B Substituted triazole derivative and application thereof in preparation of anti-tumor metastasis drugs 浙江大学 2020-01-21 CN disclosed
CN-108191781-A Substituted 1,2,4-triazole analog derivative and its application in medicine for anti transfer of tumor is prepared 浙江大学 2018-06-22 CN disclosed