SCHEMBL2828042

SCHEMBL2828042

Cc1nc2c(N3CCC(O)(c4ccccc4)CC3)cccc2c(-c2ccccc2)c1C(=O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MCHR1 Q99705 3/20 0.37
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
MLYCD O95822 1/20 0.35
TACR1 P25103 2/20 0.35
SCN9A Q15858 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
RPS6KB1 P23443 1/20 0.34
RBP4 P02753 1/20 0.34
TTR P02766 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828013 0.95 ALDH1A1 (0.36) MAPTMCHR1ALDH1A1MLYCD
SCHEMBL2825542 0.92 KIF18A (0.35) MCHR1ALDH1A1MEN1KMT2APDE4B
SCHEMBL2824028 0.87 FABP3 (0.43) MAPTSMN1; SMN2GAANPSR1ALDH1A1
SCHEMBL2825677 0.86 FABP3 (0.45) MAPTSMN1; SMN2GAANPSR1ALDH1A1
SCHEMBL2821880 0.86 FABP3 (0.45) MAPTSMN1; SMN2GAANPSR1ALDH1A1
SCHEMBL2826514 0.85 TACR1 (0.42) MAPTSMN1; SMN2GAANPSR1POLB
SCHEMBL2826068 0.85 NPSR1 (0.43) MAPTSMN1; SMN2GAANPSR1ALDH1A1
SCHEMBL2823196 0.82 GAA (0.40) MAPTSMN1; SMN2NPC1RAB9AGAA
SCHEMBL2821958 0.81 FABP3 (0.43) MAPTSMN1; SMN2NPC1RAB9AMCHR1
SCHEMBL2821151 0.80 KIF18A (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed