SCHEMBL28232171

SCHEMBL28232171

Cc1c(F)c(F)c(-c2cccc3ccccc23)c(F)c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.47
CYP2A6 P11509 3/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 3/20 0.41
CYP1A2 P05177 1/20 0.41
KDM4E B2RXH2 4/20 0.40
TYMP P19971 1/20 0.39
GSK3B P49841 1/20 0.39
ADK P55263 1/20 0.39
ENPP3 O14638 1/20 0.38
ENPP1 P22413 1/20 0.38
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP1 P29466 1/20 0.37
RAB9A P51151 1/20 0.37
CASP7 P55210 1/20 0.37
ATM Q13315 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138564 0.88 DHFR (0.44) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL26750936 0.86 DHFR (0.43) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL26750829 0.82 DHFR (0.41) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL1455734 0.79 DHFR (0.53) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL28112434 0.78 HPRT1 (0.42) DHFRCYP2A6ALDH1A1TSHRKDM4E
SCHEMBL29892469 0.77 ALDH1A1 (0.48) CYP2A6ALDH1A1TSHRCYP1A2KDM4E
SCHEMBL27263879 0.76 ALDH1A1 (0.53) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL15856404 0.76 CYP2A6 (0.58) DHFRCYP2A6ALDH1A1TSHRCYP1A2
SCHEMBL24254765 0.76 AKR1C3 (0.39) DHFRCYP2A6ALDH1A1TSHRKDM4E
SCHEMBL15856479 0.76 ALDH1A1 (0.52) DHFRCYP2A6ALDH1A1TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106146454-B The method that Negishi couplings prepare polyfluoro biaryl hydrocarbon compound 陕西师范大学 2018-08-24 CN disclosed