SCHEMBL4138564

SCHEMBL4138564

Fc1c(F)c(F)c(-c2cccc3ccccc23)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.44
TYMP P19971 1/20 0.43
ALDH1A1 P00352 5/20 0.42
TSHR P16473 4/20 0.42
HSD17B10 Q99714 4/20 0.42
CYP2A6 P11509 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 2/20 0.40
PTPN1 P18031 1/20 0.40
ALPL P05186 1/20 0.40
GAA P10253 1/20 0.40
DNMT1 P26358 1/20 0.39
HPGD P15428 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
KEAP1 Q14145 1/20 0.39
GSK3B P49841 1/20 0.39
ADK P55263 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
HPRT1 P00492 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24254765 0.86 AKR1C3 (0.39) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL29892469 0.83 ALDH1A1 (0.48) ALDH1A1TSHRHSD17B10CYP2A6TDP1
SCHEMBL2709174 0.81 CES1 (0.41) ALDH1A1TSHRHSD17B10CYP2A6KDM4E
SCHEMBL17739662 0.80 AKR1C3 (0.36) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL29407412 0.80 ALDH1A1 (0.50) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL702934 0.80 ALDH1A1 (0.50) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL7719797 0.78 DNMT1 (0.46) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL22978397 0.78 NPC1 (0.43) DHFRTYMPALDH1A1TSHRHSD17B10
SCHEMBL13878089 0.78 KEAP1 (0.50) ALDH1A1TSHRHSD17B10TDP1KDM4E
SCHEMBL31415913 0.78 HPRT1 (0.50) DHFRTYMPALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION AOC2, AOC3, DBH DHFR 1817/4885TYMP 4670/4885ALDH1A1 44/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.