SCHEMBL28239231

SCHEMBL28239231

COc1ccc2c(c1)C(N)CN(CC(F)(F)F)C2C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.36
OPRD1 P41143 2/20 0.35
OPRK1 P41145 1/20 0.35
TIPARP Q7Z3E1 1/20 0.33
KDM1A O60341 1/20 0.33
IDH1 O75874 1/20 0.33
NQO2 P16083 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
HTR2A P28223 3/20 0.33
BRD4 O60885 1/20 0.33
DRD1 P21728 1/20 0.33
CPS1 P31327 1/20 0.32
KYAT1 Q16773 1/20 0.32
KYAT3 Q6YP21 1/20 0.32
AADAT Q8N5Z0 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
DPP4 P27487 1/20 0.32
DPP9 Q86TI2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28240049 0.85 GRIN2B (0.36) OPRM1OPRD1OPRK1TIPARPIDH1
SCHEMBL28239143 0.75 DRD1 (0.50) DRD1HTR2C
SCHEMBL1686619 0.64 KDM1A (0.42) KDM1AMTNR1AMTNR1BHTR2AKYAT1
SCHEMBL1686616 0.64 KDM1A (0.42) KDM1AMTNR1AMTNR1BHTR2AKYAT1
SCHEMBL1686617 0.64 KDM1A (0.42) KDM1AMTNR1AMTNR1BHTR2AKYAT1
SCHEMBL16624303 0.62 SLC6A2 (0.62) OPRM1DRD1KYAT1KYAT3AADAT
SCHEMBL26939190 0.62 HTR2C (0.49) OPRM1OPRD1KDM1AMTNR1AMTNR1B
SCHEMBL23929133 0.62 DRD2 (0.41) DRD1
SCHEMBL21670710 0.61 DRD2 (0.45) IDH1
SCHEMBL22970938 0.61 MAOA (0.57) BRD4DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903310-B Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain 阵列生物制药公司 2018-08-14 CN disclosed