SCHEMBL28239703

SCHEMBL28239703

[CH2]Cc1nnc(C2CCNCC2)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
HPGDS O60760 1/20 0.32
HTR2C P28335 3/20 0.32
HRH3 Q9Y5N1 1/20 0.32
SLC18A3 Q16572 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
GABRA1 P14867 3/20 0.31
GABRB2 P47870 3/20 0.31
PARP1 P09874 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
MAPK13 O15264 1/20 0.30
RAF1 P04049 1/20 0.30
MAPK9 P45984 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25919952 0.79 SLC18A3 (0.38) ADORA2AADORA2BHPGDSHTR2CHRH3
SCHEMBL27323115 0.76 CACNA1H (0.40) HRH3
SCHEMBL3949876 0.73 GABRA1 (0.52) HPGDSHTR2CSLC18A3SIGMAR1GABRA1
SCHEMBL18814355 0.72 HTR2C (0.37) ADORA2AADORA2BHPGDSHTR2CHRH3
Hydrochloric Acid SCHEMBL2902954 0.71 HTR2C (0.39) ADORA2AADORA2BHPGDSHTR2CHRH3
Hydrochloric Acid SCHEMBL31583308 0.70 HTR6 (0.46) HTR2CGABRA1GABRB2
SCHEMBL2755238 0.70 SLC6A2 (0.59) HPGDSSLC18A3SIGMAR1
Hydrochloric Acid SCHEMBL240186 0.69 SLC6A2 (0.58) HPGDSSLC18A3SIGMAR1
SCHEMBL25934002 0.68 HTR2C (0.41) HPGDSHTR2CPARP1MEN1KMT2A
SCHEMBL4796049 0.65 PARP1 (0.41) PARP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108430991-A CGRP receptor antagonist 赫普塔瑞斯医疗有限公司 2018-08-21 CN disclosed