SCHEMBL2823977

SCHEMBL2823977

CC(C)(C)c1ccc(CNC(=O)Nc2cccc(CCNC(=O)O)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.54
NPC1 O15118 5/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TRPV1 Q8NER1 2/20 0.53
CNR1 P21554 2/20 0.53
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
TP53 P04637 1/20 0.51
HPGD P15428 1/20 0.51
NR1H4 Q96RI1 1/20 0.50
MAPT P10636 3/20 0.49
ALDH1A1 P00352 1/20 0.49
ESRRG P62508 1/20 0.49
LMNA P02545 2/20 0.48
MTOR P42345 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2824601 0.88 NPC1 (0.61) RAB9ANPC1SMN1; SMN2CNR1MEN1
SCHEMBL1206065 0.86 TRPV1 (0.55) RAB9ANPC1SMN1; SMN2TRPV1CNR1
SCHEMBL2853369 0.85 RAB9A (0.65) RAB9ANPC1SMN1; SMN2CNR1MEN1
SCHEMBL12069954 0.83 NPC1 (0.78) RAB9ANPC1SMN1; SMN2TRPV1MEN1
SCHEMBL1206058 0.83 TRPV1 (0.49) RAB9ANPC1SMN1; SMN2TRPV1MEN1
SCHEMBL2827311 0.80 KMT2A (0.72) RAB9ANPC1SMN1; SMN2CNR1MEN1
SCHEMBL14860031 0.80 MTOR (0.72) RAB9ANPC1SMN1; SMN2TRPV1CNR1
SCHEMBL13167593 0.79 TRPV1 (0.71) RAB9ANPC1SMN1; SMN2TRPV1MEN1
SCHEMBL2849248 0.79 MEN1 (0.62) RAB9ANPC1SMN1; SMN2CNR1MEN1
SCHEMBL2823579 0.79 KMT2A (0.60) RAB9ANPC1SMN1; SMN2CNR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed