SCHEMBL2853369

SCHEMBL2853369

O=C(O)NCCc1cccc(NC(=O)NCc2ccc(F)cc2)c1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.65
NPC1 O15118 5/20 0.65
POLB P06746 2/20 0.65
MAOB P27338 1/20 0.65
SMN1; SMN2 Q16637 3/20 0.61
GAA P10253 1/20 0.59
CHEK1 O14757 1/20 0.54
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
MAPT P10636 2/20 0.52
CNR1 P21554 2/20 0.52
NAMPT P43490 1/20 0.52
TP53 P04637 1/20 0.51
HPGD P15428 1/20 0.51
LMNA P02545 1/20 0.51
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2824601 0.91 NPC1 (0.61) RAB9ANPC1POLBMAOBSMN1; SMN2
SCHEMBL1205503 0.85 RAB9A (0.67) RAB9ANPC1POLBMAOBSMN1; SMN2
SCHEMBL2823977 0.85 RAB9A (0.54) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL2827311 0.83 KMT2A (0.72) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL2849248 0.82 MEN1 (0.62) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL2823579 0.81 KMT2A (0.60) RAB9ANPC1POLBSMN1; SMN2KMT2A
SCHEMBL7420189 0.80 RAB9A (1.00) RAB9ANPC1POLBMAOBSMN1; SMN2
SCHEMBL8059186 0.80 KMT2A (0.55) RAB9ANPC1MAOBSMN1; SMN2GAA
SCHEMBL1205961 0.79 SMN1; SMN2 (0.56) RAB9ANPC1POLBMAOBSMN1; SMN2
SCHEMBL8176987 0.79 LMNA (0.71) RAB9ANPC1POLBMAOBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254860-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR Almirall, S.A. (ES) 2010-12-01 EP disclosed
WO-2009106351-A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL) PHENOL AS AGONISTS OF THE B2 ADRENERGIC RECEPTOR ALMIRALL, S.A. (ES) 2009-09-03 WO disclosed
EP-2096105-A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor Laboratorios Almirall, S.A. (ES) 2009-09-02 EP disclosed