SCHEMBL2823282

SCHEMBL2823282

Cc1nc2c(OC(F)(F)F)cccc2c(-c2ccc(F)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 2/20 0.39
DHODH Q02127 1/20 0.37
TNKS O95271 2/20 0.37
TNKS2 Q9H2K2 2/20 0.37
PARP2 Q9UGN5 2/20 0.37
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADORA2B P29275 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825609 0.92 SMN1; SMN2 (0.44) DHODHADORA2AADORA1ALDH1A1SMN1; SMN2
SCHEMBL2824252 0.91 FABP3 (0.38) DHODHTNKSTNKS2PARP2ADORA2A
SCHEMBL2826082 0.90 ENPP1 (0.43) ENPP1TNKSTNKS2PARP2ADORA2A
SCHEMBL2824206 0.89 DHODH (0.37) DHODHADORA2AADORA1ALDH1A1L3MBTL1
SCHEMBL2825639 0.89 NR1H2 (0.40) PTGDR2
SCHEMBL2826114 0.87 CYP1A2 (0.39) DHODHTNKSTNKS2PARP2ALDH1A1
SCHEMBL2821965 0.85 FABP3 (0.39) ADORA2AADORA1SMN1; SMN2PTGDR2KMT2A
SCHEMBL2829123 0.84 ENPP1 (0.40) ENPP1DHODHTNKSTNKS2PARP2
SCHEMBL2824267 0.82 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL2824685 0.81 KDM4E (0.41) DHODHTNKSTNKS2PARP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed