SCHEMBL2825639

SCHEMBL2825639

Cc1nc2c(OC(F)(F)F)cccc2c(-c2ccc(S(C)(=O)=O)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.40
RORC P51449 2/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
NR1H3 Q13133 1/20 0.37
PTGS2 P35354 6/20 0.36
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823282 0.89 ENPP1 (0.39) PTGDR2
SCHEMBL2825609 0.87 SMN1; SMN2 (0.44) NR1H2NR1H3
SCHEMBL2824252 0.87 FABP3 (0.38) NR1H2PTGDR2
SCHEMBL2826082 0.86 ENPP1 (0.43)
SCHEMBL2825660 0.85 NR1H2 (0.41) NR1H2NR1H3PTGS2
SCHEMBL2827841 0.85 NR1H2 (0.41) NR1H2NR1H3PTGS2PTGS1
SCHEMBL2824206 0.83 DHODH (0.37) NR1H2PTGDR2NR1H3
SCHEMBL2821965 0.81 FABP3 (0.39) PTGDR2
SCHEMBL2826114 0.80 CYP1A2 (0.39) NR1H2PTGS2PTGS1
SCHEMBL2829017 0.80 PTGS2 (0.43) NR1H2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed