SCHEMBL28243153

SCHEMBL28243153

CN1C(=O)c2ccccc2C1(C)Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 10/20 0.45
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CASP3 P42574 1/20 0.38
TTR P02766 1/20 0.37
CES1 P23141 1/20 0.37
S100A4 P26447 1/20 0.37
MDM2 Q00987 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
CACNA1B Q00975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1948836 0.80 PGR (0.47) PGRALDH1A1MEN1KMT2ACYP2D6
SCHEMBL30372076 0.73 HRH3 (0.51) PGRALDH1A1MEN1KMT2ACASP3
SCHEMBL26452862 0.72 CASP3 (0.41) PGRALDH1A1MEN1KMT2ACYP2D6
SCHEMBL22787107 0.72 PGR (0.44) PGRALDH1A1MDM2KDM4EMAPT
SCHEMBL3941349 0.72 ALDH1A1 (0.41) PGRALDH1A1MEN1KMT2ACYP2D6
SCHEMBL30620824 0.70 HRH3 (0.52) PGRALDH1A1MEN1KMT2ACASP3
SCHEMBL13136409 0.70 MDM2 (0.44) PGRALDH1A1MEN1KMT2ACYP2D6
SCHEMBL30564277 0.70 HRH3 (0.52) PGRALDH1A1MEN1KMT2ACASP3
SCHEMBL5453638 0.69 PGR (0.62) PGRALDH1A1MEN1KMT2ACYP2D6
SCHEMBL3665606 0.69 HRH3 (0.40) PGRALDH1A1MEN1KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602805-A Isoindoline, azaisoindoline, indenone and the dihydro azepine indone inhibitor of MNK1 and MNK2 效应治疗股份有限公司 2018-09-28 CN disclosed