SCHEMBL2824339

SCHEMBL2824339

CC(=O)c1c(N(C)C)nc2c(Cl)cccc2c1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 5/20 0.51
FABP5 Q01469 4/20 0.51
DHODH Q02127 1/20 0.49
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
FABP3 P05413 4/20 0.43
CYP2C9 P11712 2/20 0.43
MAP2 P11137 1/20 0.40
TP53 P04637 2/20 0.40
MEN1 O00255 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2820954 0.84 ALDH1A1 (0.54) FABP4FABP5DHODHALDH1A1KDM4E
SCHEMBL14917386 0.79 FABP4 (0.79) FABP4FABP5DHODHALDH1A1KDM4E
SCHEMBL14916313 0.77 FABP4 (0.54) FABP4FABP5ALDH1A1KDM4ELMNA
SCHEMBL2824337 0.77 FABP4 (0.65) FABP4FABP5DHODHALDH1A1KDM4E
SCHEMBL14932748 0.73 ALDH1A1 (0.48) FABP4FABP5ALDH1A1KDM4ELMNA
SCHEMBL2829190 0.72 HAVCR2 (0.55) DHODHALDH1A1HSD17B10CYP2C9CYP3A4
SCHEMBL28112715 0.72 FABP4 (0.65) FABP4FABP5DHODHLMNAFABP3
SCHEMBL24122352 0.70 DHODH (0.71) FABP4FABP5DHODHLMNATSHR
SCHEMBL2826055 0.70 ALDH1A1 (0.56) FABP4ALDH1A1KDM4ELMNAHSD17B10
SCHEMBL2823585 0.68 ALDH1A1 (0.61) FABP4ALDH1A1KDM4ELMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed