SCHEMBL28248508

SCHEMBL28248508

N#Cc1cc(C#N)cc(NCc2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 3/20 0.50
PPARA Q07869 2/20 0.47
FFAR1 O14842 1/20 0.47
HDAC6 Q9UBN7 2/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
KIF11 P52732 1/20 0.46
ADRA2A P08913 1/20 0.45
CACNA1B Q00975 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ASPH Q12797 1/20 0.41
RIOX2 Q8IUF8 1/20 0.41
KDM8 Q8N371 1/20 0.41
RXRA P19793 1/20 0.41
RXRG P48443 1/20 0.41
EPHX2 P34913 1/20 0.41
EGFR P00533 1/20 0.40
LRRK2 Q5S007 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28248503 0.84 FFAR1 (0.51) VNN1FFAR1HDAC6HDAC1HDAC8
SCHEMBL6695026 0.80 HDAC1 (0.55) VNN1PPARAFFAR1HDAC6HDAC1
SCHEMBL6691557 0.80 FFAR1 (0.54) PPARAFFAR1HDAC6HDAC1ADRA2A
SCHEMBL28249055 0.79 MAPT (0.51) FFAR1KDM4E
SCHEMBL7345712 0.77 FFAR1 (0.68) PPARAFFAR1ADRA2ACACNA1B
Hydrochloric Acid SCHEMBL1854332 0.76 KIF11 (0.59) VNN1HDAC6KIF11CACNA1BEPHX2
SCHEMBL28248607 0.75 MAPT (0.55) VNN1FFAR1CACNA1BKDM4E
SCHEMBL11936090 0.73 FFAR1 (0.59) FFAR1KIF11CACNA1BEGFR
SCHEMBL5544782 0.73 FFAR1 (0.55) PPARAFFAR1HDAC6HDAC1ADRA2A
SCHEMBL6692355 0.73 ADRA2A (0.49) PPARAFFAR1ADRA2ACACNA1BEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106431989-B The aminated compounds and its preparation method and application of N- halogenated aryls substitution 云南大学 2018-10-16 CN disclosed