SCHEMBL2824927

SCHEMBL2824927

Nc1sc(C2CCC2)nc1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
PIM1 P11309 2/20 0.36
BTK Q06187 1/20 0.36
HCAR2 Q8TDS4 2/20 0.33
GLS O94925 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CAMKK2 Q96RR4 1/20 0.33
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12210066 0.81 ALDH1A1 (0.38) ALDH1A1BTKHCAR2MEN1KMT2A
SCHEMBL6504302 0.77 ALDH1A1 (0.36) ALDH1A1BTKMEN1KMT2APOLB
SCHEMBL3529066 0.77 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ATSHRPOLB
SCHEMBL6496126 0.76 RAB9A (0.39) ALDH1A1BTKMEN1KMT2AHPGD
SCHEMBL4963424 0.73 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ATSHRPOLB
SCHEMBL12210064 0.73 RBP4 (0.36) HCAR2NPC1RAB9A
SCHEMBL7995864 0.73 HCAR2 (0.35) ALDH1A1BTKHCAR2POLBNPC1
SCHEMBL21858616 0.70 ALDH1A1 (0.49) ALDH1A1BTKHCAR2KMT2ATSHR
SCHEMBL27100101 0.69 ALDH1A1 (0.36) ALDH1A1BTKMEN1KMT2APOLB
SCHEMBL15534756 0.69 COPS5 (0.39) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP disclosed