SCHEMBL2824985

SCHEMBL2824985

Cc1nc2c(N3CCOCC3)cccc2c(-c2ccc(F)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.42
TSHR P16473 2/20 0.38
AKT1 P31749 1/20 0.38
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CFTR P13569 2/20 0.37
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
PIK3CG P48736 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 2/20 0.36
RAF1 P04049 3/20 0.36
BRAF P15056 3/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826068 0.92 NPSR1 (0.43) HPGDTSHRGAAALDH1A1SMN1; SMN2
SCHEMBL2821184 0.91 SMN1; SMN2 (0.37) HPGDTSHRALDH1A1SMN1; SMN2MEN1
SCHEMBL2822062 0.90 KDM4E (0.38) HPGDTSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL2825467 0.90 KDM4E (0.38) HPGDTSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL2824314 0.85 ENPP1 (0.35) HPGDGAAALDH1A1SMN1; SMN2MEN1
SCHEMBL2824392 0.84 RAF1 (0.37) RAF1BRAF
SCHEMBL2828013 0.84 ALDH1A1 (0.36) ALDH1A1MAPT
SCHEMBL2824028 0.83 FABP3 (0.43) HPGDGAAALDH1A1SMN1; SMN2MEN1
SCHEMBL2825677 0.82 FABP3 (0.45) HPGDGAAALDH1A1SMN1; SMN2MEN1
SCHEMBL2821880 0.82 FABP3 (0.45) HPGDGAAALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed