SCHEMBL2821184

SCHEMBL2821184

Cc1nc2c(N3CCCC3)cccc2c(-c2ccc(F)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ENPP1 P22413 1/20 0.36
KCNQ2 O43526 2/20 0.36
FABP3 P05413 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
FABP4 P15090 1/20 0.36
FABP5 Q01469 1/20 0.36
MAPT P10636 2/20 0.36
DHODH Q02127 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTT P42858 2/20 0.34
REV1 Q9UBZ9 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825467 0.99 KDM4E (0.38) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2822062 0.99 KDM4E (0.38) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2824028 0.92 FABP3 (0.43) SMN1; SMN2KDM4EALDH1A1HPGDFABP3
SCHEMBL2824985 0.91 HPGD (0.42) SMN1; SMN2ALDH1A1HPGDHSD17B10MAPT
SCHEMBL2825677 0.91 FABP3 (0.45) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2821880 0.91 FABP3 (0.45) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2829017 0.88 PTGS2 (0.43) DPP4
SCHEMBL2824314 0.88 ENPP1 (0.35) SMN1; SMN2KDM4EALDH1A1HPGDENPP1
SCHEMBL2821527 0.88 PTGS2 (0.45) FABP3CYP3A4CYP2D6CYP2C9FABP4
SCHEMBL2824392 0.87 RAF1 (0.37) ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed