SCHEMBL28253155

SCHEMBL28253155

FC(F)(F)Oc1ccc(Cc2ccc(-c3ccc4ncccc4c3)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.55
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
POLB P06746 1/20 0.54
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
DYRK1A Q13627 1/20 0.46
SCN5A Q14524 2/20 0.43
CYP17A1 P05093 1/20 0.42
WNT3A P56704 1/20 0.41
GPR39 O43194 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
SCN1A P35498 1/20 0.41
SCN4A P35499 1/20 0.41
KCNH2 Q12809 1/20 0.41
SCN9A Q15858 1/20 0.41
SCN2A Q99250 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28158974 0.92 NPC1 (0.64) METNPC1RAB9APOLBCYP11B1
SCHEMBL28250224 0.91 MET (0.55) METNPC1RAB9APOLBCYP11B1
SCHEMBL30340908 0.81 NPC1 (0.60) METNPC1RAB9APOLBDYRK1A
SCHEMBL2722588 0.80 CBFB (0.52) METNPC1RAB9APOLBSCN5A
Ammonia Solution, Strong SCHEMBL11973863 0.79 CBFB (0.51) METNPC1RAB9APOLBSCN5A
SCHEMBL30340882 0.79 SCN5A (0.44) METNPC1RAB9APOLBDYRK1A
SCHEMBL1646308 0.77 TGFBR1 (0.66) MET
SCHEMBL22621116 0.77 SLC6A4 (0.51) CYP11B1CYP11B2SCN5AALDH1A1SCN1A
SCHEMBL3407902 0.76 SLC6A4 (0.49) NPC1RAB9ACYP11B1CYP11B2GPR39
SCHEMBL28172166 0.75 PDGFRB (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108697705-A combination product 利物浦热带医学院 2018-10-23 CN claimed
CN-108697705-A combination product 利物浦热带医学院 2018-10-23 CN disclosed