SCHEMBL3407902

SCHEMBL3407902

FC(F)(F)Oc1ccc(Cc2ncccn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.49
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
GPR39 O43194 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
RXRA P19793 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TLR7 Q9NYK1 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
MBOAT4 Q96T53 1/20 0.41
MPO P05164 1/20 0.41
TSHR P16473 1/20 0.41
DHODH Q02127 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2092054 0.80 SLC6A4 (0.56) SLC6A4CYP11B1CYP11B2GRIN2BALDH1A1
SCHEMBL28250224 0.79 MET (0.55) SLC6A4CYP11B1CYP11B2GPR39ALDH1A1
SCHEMBL6636466 0.78 SLC6A4 (0.52) SLC6A4CYP11B1CYP11B2GPR39TDP1
SCHEMBL16770891 0.77 SLC6A4 (0.58) SLC6A4CYP11B1CYP11B2GRIN2BALDH1A1
SCHEMBL28250250 0.77 SLC6A4 (0.51) SLC6A4CYP11B1CYP11B2GPR39MAPT
SCHEMBL28253155 0.76 MET (0.55) CYP11B1CYP11B2GPR39ALDH1A1KDM4E
SCHEMBL508197 0.76 SLC6A4 (0.49) SLC6A4CYP11B1CYP11B2GRIN2BALDH1A1
SCHEMBL28097055 0.76 LTA4H (0.59) ALDH1A1NPC1MAPTRAB9A
SCHEMBL22621116 0.75 SLC6A4 (0.51) SLC6A4CYP11B1CYP11B2ALDH1A1MPO
SCHEMBL2749763 0.74 DHODH (0.58) CYP11B1CYP11B2TDP1TLR7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114174293-A 4- (imidazo [1,2-a ] pyridin-3-yl) -pyrimidine derivatives 默克专利股份公司 2022-03-11 CN disclosed
EP-2257539-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2010-12-08 EP disclosed
WO-2009117269-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES MERCK & CO., INC. (US) 2009-09-24 WO disclosed