SCHEMBL28255602

SCHEMBL28255602

N#Cc1nc(NCc2ccccc2)c(NCc2ccccc2)nc1C#N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 9/20 0.55
GAA P10253 5/20 0.55
LMNA P02545 3/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
KDM4E B2RXH2 11/20 0.51
TSHR P16473 2/20 0.51
HSD17B10 Q99714 1/20 0.51
ALDH1A1 P00352 9/20 0.51
NPSR1 Q6W5P4 3/20 0.51
RXFP1 Q9HBX9 1/20 0.51
MAPK1 P28482 1/20 0.51
MAPT P10636 4/20 0.50
HTT P42858 3/20 0.50
CHUK O15111 1/20 0.49
KMT2A Q03164 4/20 0.49
RAD52 P43351 2/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090946 0.87 HPGD (0.55) HPGDGAALMNAL3MBTL1KDM4E
SCHEMBL28257291 0.84 LOXL2 (0.53) HPGDLMNAKDM4ETSHRHSD17B10
SCHEMBL28866282 0.82 ALDH1A1 (0.50) HPGDGAALMNAKDM4ETSHR
SCHEMBL28257132 0.82 KDM4E (0.51) HPGDGAALMNAKDM4EHSD17B10
SCHEMBL28257168 0.82 APP (0.46) HPGDGAALMNAL3MBTL1TSHR
SCHEMBL28255594 0.82 PDE4A (0.57) HPGDGAALMNAKDM4ETSHR
SCHEMBL28257164 0.80 APP (0.51) HPGDGAAL3MBTL1KDM4EALDH1A1
SCHEMBL28255597 0.80 CYP1A2 (0.52) HPGDGAALMNAL3MBTL1KDM4E
SCHEMBL26921535 0.79 HPGD (0.47) HPGDGAALMNAL3MBTL1KDM4E
SCHEMBL28255605 0.78 TSHR (0.63) HPGDGAALMNAKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929280-A Pyrazine derivative and its preparation method and pharmaceutical composition and purposes 中国医学科学院药物研究所 2018-12-04 CN claimed