SCHEMBL28255605

SCHEMBL28255605

COc1ccc(CNc2nc(C#N)c(C#N)nc2NCc2ccc(OC)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.63
MAPT P10636 9/20 0.56
GAA P10253 7/20 0.56
ALDH1A1 P00352 4/20 0.56
KDM4E B2RXH2 2/20 0.56
HPGD P15428 2/20 0.56
HSD17B10 Q99714 2/20 0.56
TP53 P04637 2/20 0.56
MAPK1 P28482 1/20 0.56
NPC1 O15118 1/20 0.54
HTT P42858 3/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
PDE5A O76074 1/20 0.52
LMNA P02545 4/20 0.52
HIF1A Q16665 1/20 0.52
GLA P06280 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4726558 0.84 TSHR (0.55) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL26921894 0.83 TSHR (0.55) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL28257291 0.80 LOXL2 (0.53) TSHRMAPTALDH1A1KDM4EHPGD
SCHEMBL28866282 0.79 ALDH1A1 (0.50) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL28257132 0.79 KDM4E (0.51) MAPTGAAALDH1A1KDM4EHPGD
SCHEMBL28257168 0.79 APP (0.46) TSHRMAPTGAAHPGDNPC1
SCHEMBL28255602 0.78 HPGD (0.55) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL23040086 0.77 TSHR (0.55) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL18953194 0.77 NPC1 (0.54) TSHRMAPTGAAALDH1A1KDM4E
SCHEMBL29499805 0.77 TSHR (0.55) TSHRMAPTGAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929280-A Pyrazine derivative and its preparation method and pharmaceutical composition and purposes 中国医学科学院药物研究所 2018-12-04 CN claimed