SCHEMBL28866282

SCHEMBL28866282

N#Cc1nc(NCc2ccc(F)cc2)c(NCc2ccc(F)cc2)nc1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 5/20 0.50
KDM4E B2RXH2 4/20 0.50
GAA P10253 4/20 0.50
HSD17B10 Q99714 3/20 0.50
MAPT P10636 7/20 0.47
NPSR1 Q6W5P4 4/20 0.47
MAPK1 P28482 2/20 0.47
TSHR P16473 1/20 0.47
ATM Q13315 1/20 0.47
LMNA P02545 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KCNH3 Q9ULD8 2/20 0.46
HTT P42858 1/20 0.46
APP P05067 1/20 0.46
CTSL P07711 3/20 0.45
KDM4C Q9H3R0 1/20 0.45
MAP2K4 P45985 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28257291 0.84 LOXL2 (0.53) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL28257168 0.83 APP (0.46) HPGDGAAMAPTTSHRLMNA
SCHEMBL28257132 0.83 KDM4E (0.51) ALDH1A1HPGDKDM4EGAAHSD17B10
SCHEMBL28255602 0.82 HPGD (0.55) ALDH1A1HPGDKDM4EGAAHSD17B10
SCHEMBL28257164 0.81 APP (0.51) ALDH1A1HPGDKDM4EGAAMAPK1
SCHEMBL28255605 0.79 TSHR (0.63) ALDH1A1HPGDKDM4EGAAHSD17B10
SCHEMBL28257153 0.78 VNN1 (0.46) GAAMAP2K4VNN1
SCHEMBL29558696 0.75 MEN1 (0.63) HPGDKDM4EMAPTNPSR1MAPK1
SCHEMBL28257188 0.73 MEN1 (0.45) ALDH1A1HPGDKDM4EGAAHSD17B10
SCHEMBL1715740 0.73 HPGD (0.51) ALDH1A1HPGDKDM4EGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108929280-A Pyrazine derivative and its preparation method and pharmaceutical composition and purposes 中国医学科学院药物研究所 2018-12-04 CN claimed