SCHEMBL2825595

SCHEMBL2825595

COc1ccc(C#Cc2cc(C#Cc3ccc(OC)c(OC)c3)cc(Sc3ccc(O)c(C)c3)c2)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.36
ACACB O00763 2/20 0.35
DHFR P00374 1/20 0.35
MAOB P27338 1/20 0.35
AR P10275 4/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
CHEK1 O14757 1/20 0.34
ACHE P22303 1/20 0.33
APP P05067 1/20 0.33
ALOX15 P16050 2/20 0.33
ALOX12 P18054 1/20 0.33
HTR1A P08908 1/20 0.32
HTR3A P46098 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
GFER P55789 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825593 0.84 ACACB (0.35) ACACBDHFRARALDH1A1MAPT
SCHEMBL2827415 0.82 GRM5 (0.44)
SCHEMBL2070877 0.77 PPARA (0.43) ACACBALDH1A1MAPTACHEALOX15
SCHEMBL29438804 0.72 TP53 (0.54) ARALDH1A1MAPTALOX15ALOX12
SCHEMBL51244 0.72 TP53 (0.54) ARALDH1A1MAPTALOX15ALOX12
SCHEMBL2820981 0.72 ERN1 (0.47)
SCHEMBL2820963 0.72 HSP90AA1 (0.32) AR
SCHEMBL18130105 0.71 APP (0.62) ACACBMAOBCHEK1ACHEAPP
SCHEMBL16641175 0.71 CA2 (0.54) ACACBARALDH1A1ACHEHTR3A
SCHEMBL10710607 0.69 NR1H2 (0.58) ARALDH1A1MAPTACHEALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed