SCHEMBL2825593

SCHEMBL2825593

COc1ccc(C#Cc2cc(C#Cc3ccc(OC)c(OC)c3)cc(Sc3ccc([O])c(C)c3)c2)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.35
DHFR P00374 3/20 0.35
AR P10275 5/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HTR1A P08908 1/20 0.34
HTR3A P46098 1/20 0.34
TYMS P04818 1/20 0.34
ACHE P22303 1/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
KDR P35968 1/20 0.33
CHEK2 O96017 1/20 0.33
TLR9 Q9NR96 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825595 0.84 P4HB (0.36) ACACBDHFRARALDH1A1MAPT
SCHEMBL2827409 0.82 GRM5 (0.47)
SCHEMBL2070877 0.77 PPARA (0.43) ACACBALDH1A1MAPTACHE
SCHEMBL2820978 0.72 GRM5 (0.44) KDR
SCHEMBL2825829 0.71 GRM5 (0.43) ACACBALDH1A1MAPT
SCHEMBL16641175 0.71 CA2 (0.54) ACACBARALDH1A1HTR3AACHE
SCHEMBL14176700 0.69 AR (0.44) ARALDH1A1MAPTACHEPDGFRB
SCHEMBL30832957 0.69 CA2 (0.52) DHFRARALDH1A1MAPTHTR1A
SCHEMBL7859196 0.69 CA2 (0.52) DHFRARALDH1A1MAPTHTR1A
SCHEMBL2821756 0.69 GRM5 (0.41) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed