SCHEMBL2827415

SCHEMBL2827415

COc1cccc(C#Cc2cc(C#Cc3cccc(OC)c3)cc(Sc3ccc(O)c(C)c3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
FFAR1 O14842 1/20 0.40
EGLN1 Q9GZT9 1/20 0.38
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
HAO1 Q9UJM8 1/20 0.37
PTPN6 P29350 1/20 0.36
PTPN11 Q06124 1/20 0.36
PTPN22 Q9Y2R2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2827409 0.85 GRM5 (0.47) GRM5CA12CA1CA2CA9
SCHEMBL2825595 0.82 P4HB (0.36)
SCHEMBL2068502 0.79 PPARD (0.53) FFAR1EGLN1
SCHEMBL2068483 0.76 MMP2 (0.41) GRM5CA12CA1CA2CA9
SCHEMBL2820981 0.75 ERN1 (0.47) GRM5FFAR1
SCHEMBL29640424 0.73 CA12 (0.59) GRM5CA12CA1CA2CA9
SCHEMBL2820963 0.72 HSP90AA1 (0.32) HSP90AA1
SCHEMBL6132140 0.72 GRM5 (0.66) GRM5CA12CA1CA2CA9
SCHEMBL30707880 0.72 GRM5 (0.66) GRM5CA12CA1CA2CA9
SCHEMBL51244 0.71 TP53 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed