SCHEMBL28256378

SCHEMBL28256378

Nc1ccc(-c2ccc(Nc3ccc(S(N)(=O)=O)cc3)cc2)cc1NC=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 5/20 0.46
CA2 P00918 12/20 0.44
CA9 Q16790 12/20 0.44
CA12 O43570 11/20 0.44
CA1 P00915 10/20 0.43
CA14 Q9ULX7 2/20 0.42
CDK1 P06493 2/20 0.42
CDK2 P24941 2/20 0.42
CCNB1 P14635 1/20 0.42
CCNA2 P20248 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA5B Q9Y2D0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779494 0.79 HDAC2 (0.43)
SCHEMBL10707842 0.76 HDAC1 (0.43)
SCHEMBL28256379 0.74 IKBKB (0.55) SOS1CA2CA9CA12CA1
SCHEMBL1414315 0.72 CA2 (0.59) CA2CA9CA12CA1CA14
SCHEMBL28107398 0.72 SOS1 (0.70) SOS1CA2CA9CA12CA1
SCHEMBL671915 0.69 CA2 (0.74) SOS1CA2CA9CA12CA1
SCHEMBL5221358 0.68 MAPT (0.61) SOS1CA2CA9CA12CA1
SCHEMBL11577144 0.67 HTR6 (0.45)
SCHEMBL16640691 0.67 IKBKB (0.57)
SCHEMBL29032711 0.67 HDAC2 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108785292-A AMINO-ARYL-BENZAMIDE COMPOUNDS AND METHODS OF USE THEREOF 上海赫普化医药技术有限公司 2018-11-13 CN disclosed