SCHEMBL2825846

SCHEMBL2825846

O=C(Nc1cccc(F)c1)Oc1ncsc1Nc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
HPGD P15428 1/20 0.46
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
ATM Q13315 1/20 0.42
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
GFER P55789 1/20 0.41
KCNK3 O14649 1/20 0.41
FAAH O00519 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829854 0.87 SMN1; SMN2 (0.44) KMT2ANPC1RAB9ALMNAKDM4E
SCHEMBL2830000 0.87 NPC1 (0.47) KMT2AMEN1NPC1RAB9AHPGD
SCHEMBL2827687 0.86 MEN1 (0.49) KMT2AMEN1NPC1RAB9AHPGD
SCHEMBL2828100 0.85 NPC1 (0.46) KMT2AMEN1NPC1RAB9AHPGD
SCHEMBL2825247 0.83 NPC1 (0.44) KMT2AMEN1NPC1RAB9ALMNA
SCHEMBL2828853 0.82 KMT2A (0.43) KMT2AMEN1NPC1RAB9AKDM4E
SCHEMBL2826737 0.82 RAB9A (0.56) KMT2AMEN1NPC1RAB9ATP53
SCHEMBL2828482 0.81 NPC1 (0.50) KMT2AMEN1NPC1RAB9ATP53
SCHEMBL2830058 0.81 LMNA (0.50) KMT2AMEN1NPC1RAB9AHPGD
SCHEMBL2827177 0.78 ALDH1A1 (0.46) KMT2AMEN1LMNACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed