SCHEMBL28258654

SCHEMBL28258654

O=CNc1ccc2c(NC=O)n[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 7/20 0.41
DYRK1A Q13627 4/20 0.40
MAPK10 P53779 1/20 0.39
MAPK14 Q16539 1/20 0.39
MAP2K4 P45985 1/20 0.38
GSK3B P49841 4/20 0.37
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
KCNQ1 P51787 1/20 0.36
SCN5A Q14524 1/20 0.36
AAK1 Q2M2I8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91462 0.78 DYRK1A (0.40) DYRK1AMAP2K4GSK3B
SCHEMBL11754096 0.77 TRPA1 (0.50) TRPA1MAPK10MAP2K4
SCHEMBL28079409 0.76 TRPA1 (0.49) TRPA1MAPK10MAP2K4
Hydrochloric Acid SCHEMBL8487463 0.76 TRPA1 (0.49) TRPA1MAPK10MAP2K4
SCHEMBL11755947 0.73 JAK2 (0.54) DYRK1A
SCHEMBL28972793 0.73 HDAC6 (0.60) GSK3B
SCHEMBL25200397 0.72 PDPK1 (0.53) DYRK1AMAPK10MAPK14GSK3B
SCHEMBL11748390 0.72 FADS1 (0.54) TRPA1MAP2K4GSK3BKCNQ3KCNQ2
SCHEMBL11748510 0.69 NTRK1 (0.43) MAPK10GSK3B
SCHEMBL26393980 0.69 GSK3B (0.57) DYRK1AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109121414-A Benzopyrazole compounds and analogs thereof 拜奥克里斯特制药公司 2019-01-01 CN disclosed