SCHEMBL2825870

SCHEMBL2825870

Cc1nc(OC(=O)Nc2ccn(C)n2)c(Nc2ccnc(Cl)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.39
S1PR2 O95136 1/20 0.38
SMARCA2 P51531 3/20 0.38
SMARCA4 P51532 3/20 0.38
RAB9A P51151 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
MAPT P10636 1/20 0.36
GRM5 P41594 3/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
NOTUM Q6P988 1/20 0.35
MAPK1 P28482 1/20 0.35
PDE4B Q07343 1/20 0.35
PIK3CA P42336 1/20 0.35
MAPK8 P45983 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828939 0.86 SMARCA2 (0.48) NPC1SMARCA2SMARCA4RAB9AGRM5
SCHEMBL2833176 0.84 SORT1 (0.41) NPC1SMARCA2SMARCA4RAB9AMAPT
SCHEMBL2826482 0.84 NPC1 (0.40) NPC1S1PR2RAB9ASMN1; SMN2KDM4E
SCHEMBL2827627 0.83 SMARCA2 (0.43) NPC1SMARCA2SMARCA4RAB9AGRM5
SCHEMBL2831219 0.83 NPC1 (0.37) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL2827806 0.82 GRM5 (0.44) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL2826248 0.82 SMARCA2 (0.56) NPC1SMARCA2SMARCA4RAB9AGRM5
SCHEMBL2827684 0.82 GRM5 (0.48) NPC1RAB9AGRM5JAK2NOTUM
SCHEMBL2826030 0.82 PIK3CA (0.37) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL2829284 0.81 NPC1 (0.41) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed