SCHEMBL2829284

SCHEMBL2829284

Cc1nc(OC(=O)Nc2ccn(C)n2)c(Nc2cccc(CO)c2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
ABCG2 Q9UNQ0 1/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GRM5 P41594 2/20 0.36
NOTUM Q6P988 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
KCNH2 Q12809 1/20 0.35
JAK3 P52333 1/20 0.34
BTK Q06187 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
KDM1A O60341 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828971 0.91 NPC1 (0.37) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL2827914 0.85 GRM5 (0.47) NPC1RAB9AABCG2LMNASMN1; SMN2
SCHEMBL2830183 0.85 NPC1 (0.40) NPC1RAB9AABCG2ALDH1A1LMNA
SCHEMBL5197589 0.84 GRM5 (0.52) NPC1RAB9AABCG2ALDH1A1LMNA
SCHEMBL2827684 0.82 GRM5 (0.48) NPC1RAB9AGRM5NOTUMJAK3
SCHEMBL2831219 0.82 NPC1 (0.37) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL2825870 0.81 NPC1 (0.39) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL2830402 0.81 MAPT (0.45) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL2827806 0.81 GRM5 (0.44) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL2826783 0.80 GRM5 (0.49) ABCG2ALDH1A1LMNAGRM5MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed