SCHEMBL28259407

SCHEMBL28259407

O=C(O)N1CC(N2CCOc3c(F)cccc32)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.42
NOTUM Q6P988 2/20 0.36
HTR6 P50406 2/20 0.36
PIK3CB P42338 3/20 0.36
PIK3CD O00329 2/20 0.36
PIK3CG P48736 2/20 0.36
SCN9A Q15858 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 2/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
UCHL1 P09936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28261103 0.78 NOTUM (0.45) AVPR1ANOTUMSCN9AKDM4EALOX15
SCHEMBL20328102 0.77 AVPR1A (0.41) AVPR1AHTR6PIK3CBPIK3CDPIK3CG
SCHEMBL30962043 0.76 SCN9A (0.44) AVPR1ANOTUMHTR6PIK3CBPIK3CD
SCHEMBL28261074 0.74 AGTR2 (0.46) AVPR1APIK3CBPIK3CDPIK3CGALDH1A1
SCHEMBL18222113 0.74 NOTUM (0.47) NOTUMMEN1KMT2ALMNAUSP30
SCHEMBL1449558 0.73 L3MBTL3 (0.37) NOTUMKDM4EALDH1A1UCHL1USP30
SCHEMBL30962073 0.72 PIK3CD (0.38) AVPR1ANOTUMHTR6PIK3CBPIK3CD
SCHEMBL2015384 0.71 SOS1 (0.42) AVPR1AHTR6PIK3CBPIK3CDPIK3CG
SCHEMBL20328103 0.70 AVPR1A (0.54) AVPR1AKDM4EMEN1KMT2AALDH1A1
SCHEMBL1802527 0.68 ADRA2A (0.39) NOTUMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884071-B Condensed ring based azetidinyl triazole derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2021-05-14 CN disclosed
CN-108884071-A Condensed ring based azetidinyl triazole derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2018-11-23 CN disclosed