SCHEMBL28263108

SCHEMBL28263108

O=CC1CNC(c2cccc(Cl)c2)N1O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.41
HDAC2 Q92769 1/20 0.41
SLC6A2 P23975 5/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TRPM4 Q8TD43 1/20 0.36
TRPM5 Q9NZQ8 1/20 0.36
SLC6A4 P31645 1/20 0.36
GID4 Q8IVV7 1/20 0.36
CHRNA7 P36544 1/20 0.36
SLC9A1 P19634 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28263134 0.84 KDM1A (0.37) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL19328932 0.72 SLC6A3 (0.49) SLC6A3HDAC2SLC6A2KDM4EALDH1A1
SCHEMBL28263132 0.68 ABCB1 (0.44) ALDH1A1
SCHEMBL1072730 0.68 SLC6A3 (0.54) SLC6A3HDAC2SLC6A2HTR2AHTR2C
SCHEMBL20835816 0.68 FFAR2 (0.43) CHRNA7
SCHEMBL27410715 0.68 SLC6A3 (0.41) SLC6A3HDAC2SLC6A2SLC6A4GID4
SCHEMBL24738322 0.66 HTR2A (0.53) SLC6A3SLC6A2HTR2AHTR2CHTR2B
SCHEMBL2916068 0.66 HTR2A (0.53) SLC6A3SLC6A2HTR2AHTR2CHTR2B
SCHEMBL28790737 0.65 SLC6A3 (0.49) SLC6A3HDAC2SLC6A2HTR2AHTR2C
SCHEMBL27492442 0.64 HTR2C (0.53) SLC6A3SLC6A2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071457-A Inhibitors of indoleamine 2, 3-dioxygenase 荷兰转化研究中心有限责任公司 2018-12-21 CN disclosed