SCHEMBL28263132

SCHEMBL28263132

O=CC1CN(C(=O)c2ccccc2)C(c2cccc(Cl)c2)N1O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
CNR2 P34972 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
CCR5 P51681 1/20 0.39
EPHX2 P34913 1/20 0.39
RECQL P46063 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GRM5 P41594 1/20 0.39
ADAM17 P78536 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GRIN2B Q13224 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28263101 0.86 HDAC4 (0.40) ABCB1KMT2AMEN1RECQLL3MBTL1
SCHEMBL28261949 0.84 ALDH1A1 (0.46) KMT2AMEN1L3MBTL1GRM5ALDH1A1
SCHEMBL28867362 0.84 LMNA (0.37) KMT2AMEN1EPHX2L3MBTL1GRM5
SCHEMBL28263098 0.78 KMT2A (0.36) ABCB1KMT2AMEN1
SCHEMBL28263118 0.76 HSD11B1 (0.41) KMT2AMEN1ALDH1A1
SCHEMBL28261985 0.76 RORC (0.45) KMT2AMEN1EPHX2ALDH1A1
SCHEMBL19328943 0.75 MEN1 (0.47) ABCB1ABCG2CNR2KMT2AMEN1
SCHEMBL28261986 0.74 CCR5 (0.36) KMT2AMEN1CCR5L3MBTL1ALDH1A1
SCHEMBL28261971 0.73 GRM5 (0.40) CCR5EPHX2L3MBTL1GRM5ALDH1A1
SCHEMBL28261984 0.72 LMNA (0.39) KMT2AMEN1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071457-A Inhibitors of indoleamine 2, 3-dioxygenase 荷兰转化研究中心有限责任公司 2018-12-21 CN disclosed