SCHEMBL28266397

SCHEMBL28266397

Cc1[c]nnn1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 8/20 0.44
RXRA P19793 8/20 0.43
GRIN1 Q05586 8/20 0.43
GRIN2B Q13224 8/20 0.43
KCNH2 Q12809 2/20 0.43
NPY5R Q15761 1/20 0.42
PIM3 Q86V86 2/20 0.39
PIM2 Q9P1W9 2/20 0.39
MLYCD O95822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28266322 0.85 L3MBTL1 (0.44) RXRAGRIN1GRIN2B
SCHEMBL28266413 0.83 PIM1 (0.46) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL28267817 0.81 CYP1A2 (0.47) NPY5R
SCHEMBL31465861 0.75 PDE10A (0.48) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL18161248 0.72 ALDH1A1 (0.61) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL18504510 0.72 PIM1 (0.46) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL6671149 0.72 RXRA (0.41) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL28266377 0.72 RXRA (0.47) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL28459519 0.71 S1PR4 (0.45) PIM1RXRAGRIN1GRIN2BKCNH2
SCHEMBL7155477 0.70 KCNH2 (0.42) PIM1RXRAGRIN1GRIN2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071488-A Substituted 1,2,3- triazole is as NR2B- selective NMDA regulator 詹森药业有限公司 2018-12-21 CN claimed
CN-109071488-A Substituted 1,2,3- triazole is as NR2B- selective NMDA regulator 詹森药业有限公司 2018-12-21 CN disclosed