SCHEMBL7155477

SCHEMBL7155477

Cc1n[c]cn1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.42
RXRA P19793 7/20 0.40
GRIN1 Q05586 7/20 0.40
GRIN2B Q13224 7/20 0.40
PDE10A Q9Y233 1/20 0.38
DHFR P00374 1/20 0.38
PHGDH O43175 1/20 0.37
NOTUM Q6P988 1/20 0.37
GRM5 P41594 1/20 0.37
NPY5R Q15761 1/20 0.36
CCKAR P32238 1/20 0.36
PIM1 P11309 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MLYCD O95822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7155610 0.84 POLB (0.48) KCNH2RXRAGRIN1GRIN2BDHFR
SCHEMBL7154140 0.83 KCNH2 (0.47) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL8139457 0.73 KCNH2 (0.43) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL28266377 0.71 RXRA (0.47) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL28266397 0.70 PIM1 (0.44) KCNH2RXRAGRIN1GRIN2BNPY5R
SCHEMBL1344378 0.69 KCNH2 (0.40) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL3147185 0.68 GPR3 (0.50) PIM1
SCHEMBL31465861 0.68 PDE10A (0.48) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL8425506 0.68 RXRA (0.39) KCNH2RXRAGRIN1GRIN2BPDE10A
SCHEMBL12245 0.67 ACHE (0.56) KCNH2GRM5L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358165-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-05 EP disclosed
WO-2002060877-A1 IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-08 WO disclosed