SCHEMBL28267152

SCHEMBL28267152

O=C(Cl)c1cc(F)cc(Cl)c1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 5/20 0.36
CES2 O00748 3/20 0.34
CES1 P23141 2/20 0.34
ALDH1A1 P00352 1/20 0.34
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
XPO1 O14980 2/20 0.33
P2RX1 P51575 2/20 0.33
TMPRSS4 Q9NRS4 2/20 0.33
NOTUM Q6P988 1/20 0.32
HPGD P15428 1/20 0.32
TLR7 Q9NYK1 1/20 0.31
P2RX4 Q99571 1/20 0.31
P2RX7 Q99572 1/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31
KDR P35968 1/20 0.31
GPR35 Q9HC97 1/20 0.31
TRPV1 Q8NER1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28208232 0.83 CES2 (0.41) ALOX15CES2ALDH1A1RXRARXRB
SCHEMBL27835356 0.83 AKR1C4 (0.41) ALDH1A1P2RX1TMPRSS4NOTUMP2RX4
SCHEMBL27964790 0.78 CES2 (0.45) ALOX15CES2CES1ALDH1A1P2RX1
SCHEMBL8103503 0.76 CES2 (0.39) ALOX15CES2CES1ALDH1A1P2RX1
SCHEMBL27835380 0.73 CES2 (0.36) ALOX15CES2CES1ALDH1A1NOTUM
SCHEMBL28265638 0.72 NOTUM (0.42) ALOX15CES2CES1ALDH1A1NOTUM
SCHEMBL42960 0.72 DDR1 (0.44) CES2ALDH1A1P2RX1TMPRSS4HPGD
SCHEMBL20268801 0.72 ALDH1A1 (0.47) ALOX15CES2CES1ALDH1A1P2RX1
SCHEMBL27853419 0.70 NOTUM (0.44) ALOX15CES2CES1ALDH1A1NOTUM
SCHEMBL28061682 0.70 RAB9A (0.37) CES2P2RX1TMPRSS4P2RX4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109195965-A The inhibitor that WDR5 protein-protein combines 普罗佩纶治疗公司 2019-01-11 CN disclosed