SCHEMBL8103503

SCHEMBL8103503

O=C(Cl)c1cc(F)cc(Cl)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.39
CES1 P23141 4/20 0.39
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 1/20 0.39
HPGD P15428 3/20 0.35
TSHR P16473 2/20 0.33
P2RX7 Q99572 5/20 0.33
HSD17B10 Q99714 2/20 0.32
CYP3A4 P08684 2/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
CASP1 P29466 1/20 0.32
KEAP1 Q14145 1/20 0.31
P2RX1 P51575 1/20 0.31
P2RX4 Q99571 1/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27964790 0.84 CES2 (0.45) CES2CES1ALDH1A1ALOX15HPGD
SCHEMBL9844447 0.83 TSHR (0.47) CES2CES1ALDH1A1TSHRCYP3A4
SCHEMBL8574493 0.81 PARP1 (0.43) CES2CES1ALDH1A1HPGDCASP1
SCHEMBL10437029 0.81 CES2 (0.38) CES2CES1HPGDTSHRP2RX7
SCHEMBL27835380 0.79 CES2 (0.36) CES2CES1ALDH1A1ALOX15HPGD
SCHEMBL27259216 0.79 CES2 (0.36) CES2CES1ALDH1A1ALOX15
SCHEMBL1311328 0.77 ALDH1A1 (0.50) ALDH1A1HPGDTSHRHSD17B10CYP3A4
SCHEMBL28267152 0.76 ALOX15 (0.36) CES2CES1ALDH1A1ALOX15HPGD
SCHEMBL11726912 0.76 TTR (0.37) ALDH1A1ALOX15HPGDTSHRHSD17B10
SCHEMBL4514781 0.75 ALDH1A1 (0.52) CES2CES1ALDH1A1ALOX15HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104725221-B The synthetic method of the chloro-5-fluorobenzoyl chloride of a kind of 2,4-bis- ZHEJIANG BENLI CHEMICAL CO., LTD. (CN) 2016-04-27 CN claimed
CN-104211590-B The preparation method of the chloro-5-fluorobenzoyl chloride of a kind of 2,4-bis- ZHEJIANG XIANFENG SCIENCE TECHNOLOGY Co.,Ltd. (CN) 2016-01-20 CN claimed
CN-105175245-A Synthesis method of 2,4-dichloro-5-fluorobenzoyl chloride SHANDONG GUOBANG PHARMACEUTICAL CO LTD 2015-12-23 CN claimed
CN-104725221-A Method for synthesizing 2,4-dichloro-5-fluorobenzoyl ZHEJIANG BENLI CHEMICAL CO LTD 2015-06-24 CN claimed
EP-0306804-A2 Process for the preparation of substituted benzyl trichlorides BAYER AG (DE) 1989-03-15 EP claimed
CN-104725221-B The synthetic method of the chloro-5-fluorobenzoyl chloride of a kind of 2,4-bis- ZHEJIANG BENLI CHEMICAL CO., LTD. (CN) 2016-04-27 CN disclosed
CN-104725221-A Method for synthesizing 2,4-dichloro-5-fluorobenzoyl ZHEJIANG BENLI CHEMICAL CO LTD 2015-06-24 CN disclosed
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
WO-1998008839-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED THIOPHENE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed
EP-0354444-A2 Process for the introduction of fluorine on aromatic nucleus by nucleophilic exchange BAYER AG (DE) 1990-02-14 EP disclosed