SCHEMBL28268352

SCHEMBL28268352

O=C(Nc1c[nH]c2ncc[c]c12)c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 9/20 0.56
PIM1 P11309 2/20 0.50
HTT P42858 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
GAK O14976 1/20 0.50
STK16 O75716 1/20 0.50
AXL P30530 1/20 0.50
NEK2 P51955 1/20 0.50
STK3 Q13188 1/20 0.50
STK11 Q15831 1/20 0.50
BMP2K Q9NSY1 1/20 0.50
TNIK Q9UKE5 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
PIM3 Q86V86 1/20 0.49
PIM2 Q9P1W9 1/20 0.49
LMNA P02545 1/20 0.49
HIF1A Q16665 1/20 0.49
GAA P10253 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053845 0.79 AAK1 (0.70) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL7110861 0.73 AAK1 (0.72) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL1469033 0.73 AAK1 (0.59) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL7548968 0.73 AAK1 (0.62) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL6643666 0.72 LMNA (0.67) PIM1HTTHDAC3HDAC1HDAC2
SCHEMBL1468749 0.71 AAK1 (0.57) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL1467820 0.71 AAK1 (0.57) AAK1PIM1HTTHDAC3HDAC1
SCHEMBL7112349 0.71 AAK1 (1.00) AAK1PIM1HDAC3HDAC1HDAC2
SCHEMBL15643127 0.70 LMNA (0.56) PIM1HTTHDAC3HDAC1HDAC2
SCHEMBL7116964 0.70 AAK1 (1.00) AAK1PIM1HDAC1GAKSTK16

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104926810-B Pyrrolopyridine as kinase inhibitor 阵列生物制药公司 2019-02-19 CN disclosed